PGP-4008Out of stock

PGP-4008

inhibits P-glycoprotein

IWP-2Out of stock

IWP-2

2-Cyano-N-(2,5-dibromophenyl)-3-hydroxy-2-butenamideOut of stock

2-Cyano-N-(2,5-dibromophenyl)-3-hydroxy-2-butenamide

inhibitor of Btk

4-Amino-1-tert-butyl-3-(1'-naphthyl)pyrazolo[3,4-d]pyrimidineOut of stock

4-Amino-1-tert-butyl-3-(1′-naphthyl)pyrazolo[3,4-d]pyrimidine

inhibitor of v-Src, c-Fyn, c-Ab

[4-tert-Butylphenyl]-N-(4-imidazol-1-yl phenyl)sulfonamideOut of stock

[4-tert-Butylphenyl]-N-(4-imidazol-1-yl phenyl)sulfonamide

c-kit activity inhibitor

N-(3,4-Dimethylphenyl)-N,4-dimethyl-benzenesulfonamide

N-(3,4-Dimethylphenyl)-N,4-dimethyl-benzenesulfonamide

A-803467

A-803467

Selective blocker of NaV1.8 channels (IC50 values are 8, 2450, 6740, 7340 and 7380 nM for hNaV1.8, hNaV1.3, hNaV1.7, hNaV1.5 and hNaV1.2 channels respectively). Shows no significant activity against T

RPV1, P2X2/3, CaV2.2 and KCNQ2/3 channels. Antinociceptive; potently attenuates mechanical allodynia in two models of neuropathic pain following i.p. administration.

MSDS UN168

CoA UN168

Mecamylamine hydrochlorideOut of stock

Mecamylamine hydrochloride

Bepridil hydrochlorideOut of stock

Bepridil hydrochloride

calcium channel blocker